Cart
sales@molnova.com
PKC-theta inhibitor
CAS No. 736048-65-0
PKC-theta inhibitor( —— )
Catalog No. M20187 CAS No. 736048-65-0
PKC-theta inhibitor is PKC-θinhibitor with an?IC50?of 12 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 239 | In Stock |
|
| 10MG | 381 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NamePKC-theta inhibitor
-
NoteResearch use only, not for human use.
-
Brief DescriptionPKC-theta inhibitor is PKC-θinhibitor with an?IC50?of 12 nM.
-
DescriptionPKC-theta inhibitor is PKC-θinhibitor with an?IC50?of 12 nM.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayAngiogenesis
-
TargetPKC
-
RecptorPKCθ
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number736048-65-0
-
Formula Weight454.4
-
Molecular FormulaC20H25F3N6O3
-
Purity>98% (HPLC)
-
SolubilityDMSO:62.5 mg/mL?(137.53 mM)
-
SMILESNCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
-
Chemical NameN4-((4-(aminomethyl)cyclohexyl)methyl)-5-nitro-N2-(2-(trifluoromethoxy)benzyl)pyrimidine-24-diamine
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Cywin CL et al. Discovery of potent and selective PKC-theta inhibitors. Bioorg Med Chem Lett. 2007 Jan 1;17(1):225-30.
molnova catalog
related products
-
p32 Inhibitor M36
p32 inhibitor M36 (M36) is a p32 mitochondrial protein inhibitor, which binds directly to p32 and inhibits p32 association with LyP-1.
-
CGP-53353
CGP-53353 (DAPH-7) is a selective inhibitor of PKCβII with IC50 of 0.41 uM, shows weak activity on PKCβI with IC50 of 3.8 uM.
-
Psychosine
Psychosine (Galactosylsphingosine) is a PKC inhibitor, a substrate for the enzyme galactosylceramide cerebrosidase (GALC), and a potential biomarker of Krabbe's disease.
